SCHEMBL7706909

SCHEMBL7706909

N#Cc1cc2cc(F)c(F)cc2o1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.52
TRPV4 Q9HBA0 2/20 0.32
GPR35 Q9HC97 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17182450 0.85 CYP2A6 (0.46) CYP2A6
SCHEMBL17182542 0.85 CYP2A6 (0.46) CYP2A6
SCHEMBL20559975 0.76 CYP2A6 (0.58) CYP2A6GPR35
SCHEMBL1995148 0.73 CYP2A6 (0.71) CYP2A6GPR35
SCHEMBL15888126 0.71 CYP2A6 (0.52) CYP2A6GPR35
SCHEMBL12321281 0.71 CYP2A6 (0.52) CYP2A6GPR35
SCHEMBL6014124 0.69 CYP2A6 (0.60) CYP2A6GPR35
SCHEMBL11550694 0.69 CYP2A6 (0.60) CYP2A6
SCHEMBL846924 0.68 CYP2A6 (1.00) CYP2A6GPR35
SCHEMBL21688675 0.68 CYP2A6 (0.58) CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906301-B1 BENZOFURYL DERIVATIVES AND THEIR USE HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
US-5955495-A BENZOFURAN-2-CARBOXAMIDINE OR 2-CARBOXAMIDOXIME COMPOUNDS USEFUL IN THE CONTROL OR PREVENTION OF ILLNESSES OR DISORDERS OF THE CENTRAL NERVOUS SYSTEM SUCH AS MIGRAINE, SCHIZOPHRENIA, ANXIETY STATES, SLEEP DISORDERS, ANOREXIA, ALZHEIMER'S HOFFMANN-LA ROCHE INC. (US) 1999-09-21 US disclosed
EP-0906301-A1 BENZOFURYL DERIVATIVES AND THEIR USE F. HOFFMANN-LA ROCHE AG (CH) 1999-04-07 EP disclosed
WO-1997042183-A1 BENZOFURYL DERIVATIVES AND THEIR USE F. HOFFMANN-LA ROCHE AG (CH) 1997-11-13 WO disclosed