SCHEMBL770786

SCHEMBL770786

c1ccc(Nc2ncc[nH]2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 6/20 0.56
ADRA2C P18825 5/20 0.56
ADRA1D P25100 3/20 0.56
ADRA1A P35348 3/20 0.56
ADRA1B P35368 3/20 0.56
TAAR1 Q96RJ0 3/20 0.52
MTOR P42345 1/20 0.47
ADK P55263 1/20 0.47
NISCH Q9Y2I1 1/20 0.47
HSD17B10 Q99714 2/20 0.46
CSNK2A1 P68400 2/20 0.46
TTBK1 Q5TCY1 1/20 0.44
TTBK2 Q6IQ55 1/20 0.44
MAPK1 P28482 2/20 0.44
ALDH1A1 P00352 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
ALOX12 P18054 1/20 0.44
PTGS1 P23219 1/20 0.44
SLC6A2 P23975 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046796 0.98 ADRA2A (0.55) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL28046706 0.98 ADRA2A (0.55) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL28046710 0.98 ADRA2A (0.55) ADRA2AADRA2CADRA1DADRA1AADRA1B
Piperazine SCHEMBL4470404 0.91 ADRA2A (0.49) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL21067687 0.86 ADRA2A (0.63) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL14629679 0.79 ADRA2A (0.56) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL5851701 0.79 ADRA2A (0.56) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL1842264 0.79 ADRA2A (0.56) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL708660 0.78 ADRA2A (0.56) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL17213665 0.77 KDM4E (0.56) ADRA2AADRA2CADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 120 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821585-B1 USE OF ALPHA 1L-AGONISTS IN THE TREATMENT OF URINARY INCONTINENCE BOEHRINGER INGELHEIM PHARMA (DE) 2007-01-10 EP claimed
EP-1285653-A1 Use of alpha-1L agonists in the treatment of incontinence Boehringer Ingelheim Pharma KG (DE) 2003-02-26 EP claimed
JP-3379960-B2 2003-02-24 JP claimed
EP-0821585-A1 USE OF $g(a) 1L? AGONISTS IN THE TREATMENT OF INCONTINENCE BOEHRINGER INGELHEIM KG (DE) 1998-02-04 EP claimed
WO-1996032939-A1 USE OF α1L AGONISTS IN THE TREATMENT OF INCONTINENCE BOEHRINGER INGELHEIM KG (DE) 1996-10-24 WO claimed
EP-0538262-A1 N-DIMETHOXY PHENYL ALKYL-N'-IMIDAZOLYL PHENYL AMIDINE DERIVATIVES AND PROCESS THEREOF IL YANG PHARM. CO., LTD. (KR) 1993-04-28 EP claimed
WO-1992000966-A1 N-DIMETHOXY PHENYL ALKYL-N'-IMIDAZOLYL PHENYL AMIDINE DERIVATIVES AND PROCESS THEREOF IL YANG PHARM. CO., LTD. (KR) 1992-01-23 WO claimed
EP-0013252-B1 CARDIAC RHYTHM REDUCTION AGENT C.H. BOEHRINGER SOHN (DE) 1987-09-23 EP claimed
EP-0029505-B1 SUBSTITUTED PHENYLAMINO-2-IMIDAZOLINE-2 DERIVATIVES, THEIR ACID ADDITION SALTS, MEDICAMENTS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION C.H. BOEHRINGER SOHN (DE) 1984-09-12 EP claimed
EP-0030620-B1 SUBSTITUTED 2-PHENYLAMINO-2-IMIDAZOLINES, ACID ADDITION SALTS THEREOF, MEDICAMENTS CONTAINING THEM AND PROCESS FOR PREPARING THEM C.H. BOEHRINGER SOHN (DE) 1984-06-13 EP claimed
EP-0007986-B1 SUBSTITUTED 2-PHENYLAMINO-IMIDAZOLINES-(2), THEIR ACID ADDITION SALTS, MEDICAMENTS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION C.H. BOEHRINGER SOHN (DE) 1981-09-16 EP claimed
EP-0031429-A1 2-(N-(2-Fluoro-6-bromophenyl)-N-(thiemyl-2-methyl)-amino)-2-imidazoline, its addition salts, pharmaceutical compositions containing them and processes for their preparation C.H. BOEHRINGER SOHN (DE) 1981-07-08 EP claimed
EP-0030620-A2 Substituted 2-phenylamino-2-imidazolines, acid addition salts thereof, medicaments containing them and process for preparing them C.H. BOEHRINGER SOHN (DE) 1981-06-24 EP claimed
EP-0030616-A1 Substituted 2-phenylamino-2-imidazolines, their acid addition salts, medicaments containing them and processes for preparing same C.H. BOEHRINGER SOHN (DE) 1981-06-24 EP claimed
EP-0029505-A1 Substituted phenylamino-2-imidazoline-2 derivatives, their acid addition salts, medicaments containing them and process for their preparation C.H. BOEHRINGER SOHN (DE) 1981-06-03 EP claimed
EP-0007991-A1 Substituted 2-phenylamino-imidazolines-(2), their acid addition salts, medicaments containing them and processes for their preparation C.H. BOEHRINGER SOHN (DE) 1980-02-20 EP claimed
EP-0007406-A1 Substituted 2-phenylamino-imidazolines-(2), their acid addition salts, medicaments containing them and processes for their preparation C.H. BOEHRINGER SOHN (DE) 1980-02-06 EP claimed
EP-0007422-A1 Substituted 2-phenylamino-imidazolines-(2), their acid addition salts, medicaments containing them and processes for their preparation C.H. BOEHRINGER SOHN (DE) 1980-02-06 EP claimed
EP-0007428-A1 Substituted 2-phenylamino-imidazolines-(2), their acid addition salts, medicaments containing them and processes for their preparation C.H. BOEHRINGER SOHN (DE) 1980-02-06 EP claimed
EP-0007438-A1 Substituted 2-phenylamino-2-imidazolines, their acid addition salts, pharmaceutical compositions containing them and process for their preparation C.H. BOEHRINGER SOHN (DE) 1980-02-06 EP claimed