SCHEMBL7707988

SCHEMBL7707988

C/C=C/C(=O)[C@H]1CC[C@H](c2cccnc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.50
HSD11B1 P28845 2/20 0.45
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
DPP4 P27487 1/20 0.41
DPP8 Q6V1X1 1/20 0.41
DPP9 Q86TI2 1/20 0.41
TNKS O95271 1/20 0.40
NAMPT P43490 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
KDM4E B2RXH2 3/20 0.39
CYP3A4 P08684 1/20 0.39
THRB P10828 1/20 0.39
TSHR P16473 1/20 0.39
THPO P40225 1/20 0.39
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL27888256 0.77 CYP11B2 (0.65) CYP11B2HSD11B1ALDH1A1L3MBTL1TNKS
SCHEMBL990213 0.76
SCHEMBL29848157 0.76
SCHEMBL7710964 0.76 KDM4E (0.35) ALDH1A1NAMPTKDM4ETSHRKMT2A
SCHEMBL7712965 0.75 KDM5A (0.37)
Formaldehyde SCHEMBL28570916 0.75 CYP11B2 (0.71) CYP11B2ALDH1A1L3MBTL1TNKSCHRNB2
SCHEMBL7704805 0.75 HCRTR2 (0.38) ALDH1A1L3MBTL1KDM4EMEN1KMT2A
Ammonia Solution, Strong SCHEMBL28985148 0.75 CYP11B2 (0.77) CYP11B2ALDH1A1CHRNB2CHRNA4MEN1
SCHEMBL2546843 0.74 CYP11B2 (0.53) CYP11B2HSD11B1ALDH1A1L3MBTL1DPP4
SCHEMBL2546841 0.74 CYP11B2 (0.53) CYP11B2HSD11B1ALDH1A1L3MBTL1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011131596-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES AS VASOPRESSIN V1A RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-10-27 WO disclosed