SCHEMBL7708154

SCHEMBL7708154

CC1Oc2ccc(CCN(Cc3cccc(Cl)c3)C(=O)OC(C)(C)C)cc2NC1=O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.44
KDR P35968 1/20 0.39
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HDAC1 Q13547 1/20 0.36
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SMYD3 Q9H7B4 1/20 0.35
RIPK1 Q13546 1/20 0.34
SLC2A1 P11166 1/20 0.34
LPAR1 Q92633 1/20 0.34
LPAR5 Q9H1C0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711139 0.94 PARP1 (0.48) PARP1KDRALDH1A1TSHRALOX15
SCHEMBL6302723 0.93 PARP1 (0.47) PARP1KDRALDH1A1TSHRALOX15
SCHEMBL7705076 0.91 HDAC1 (0.35) PARP1ALDH1A1TSHRHDAC1SMN1; SMN2
SCHEMBL7713340 0.86 PARP1 (0.47) PARP1ALDH1A1TSHRALOX15HSD17B10
SCHEMBL6308969 0.85 PARP1 (0.46) PARP1KDRALDH1A1ALOX15HSD17B10
SCHEMBL6302996 0.85 PARP1 (0.43) PARP1KDRALDH1A1TSHRALOX15
SCHEMBL6305893 0.85 PARP1 (0.54) PARP1ALDH1A1ALOX15HSD17B10HDAC1
SCHEMBL7713376 0.85 PARP1 (0.56) PARP1ALDH1A1ALOX15HSD17B10HDAC1
SCHEMBL7708255 0.84 RIPK1 (0.36) PARP1KDRTSHRALOX15HSD17B10
SCHEMBL6428132 0.83 RIPK1 (0.36) PARP1KDRTSHRALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed