SCHEMBL7708255

SCHEMBL7708255

CC1Oc2ccc(CN(Cc3cccc(Cl)c3)C(=O)OC(C)(C)C)cc2NC1=S

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.36
PARP1 P09874 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
GHSR Q92847 4/20 0.34
HSD17B10 Q99714 2/20 0.33
KDR P35968 1/20 0.33
TSHR P16473 1/20 0.33
ALOX15 P16050 1/20 0.33
CTSL P07711 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.33
SLC2A1 P11166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6428132 0.99 RIPK1 (0.36) RIPK1PARP1HDAC3HDAC1HDAC2
SCHEMBL7705076 0.94 HDAC1 (0.35) RIPK1PARP1HDAC3HDAC1HDAC2
SCHEMBL6302929 0.91 PARP1 (0.35) PARP1HDAC3HDAC1HDAC2NCOR2
SCHEMBL6309909 0.91 HSD17B10 (0.33) PARP1HDAC3HDAC1HDAC2NCOR2
SCHEMBL6309617 0.91 HDAC1 (0.43) PARP1HDAC3HDAC1HDAC2NCOR2
SCHEMBL7704945 0.91 HDAC3 (0.44) PARP1HDAC3HDAC1HDAC2NCOR2
SCHEMBL7711139 0.90 PARP1 (0.48) RIPK1PARP1HDAC3HDAC1HDAC2
SCHEMBL6302723 0.89 PARP1 (0.47) RIPK1PARP1HDAC3HDAC1HDAC2
SCHEMBL7712797 0.89 RIPK1 (0.36) RIPK1PARP1HDAC3HDAC1HDAC2
SCHEMBL7704916 0.89 HSD17B10 (0.35) PARP1SMN1; SMN2HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed