SCHEMBL7708173

SCHEMBL7708173

CC1Oc2ccc(C(C)(NC(=O)OC(C)(C)C)c3cccnc3)cc2NC1=O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PARP1 P09874 5/20 0.38
SMYD3 Q9H7B4 3/20 0.37
PDE3B Q13370 2/20 0.37
PDE3A Q14432 2/20 0.37
NAMPT P43490 2/20 0.36
RAB9A P51151 1/20 0.35
KDR P35968 1/20 0.34
CYP17A1 P05093 3/20 0.34
CYP19A1 P11511 3/20 0.34
MAOB P27338 1/20 0.33
ADORA2A P29274 1/20 0.33
RORC P51449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7093805 0.90 NAMPT (0.36) MAPTTSHRHSD17B10NAMPTRAB9A
SCHEMBL7711103 0.89 SMYD3 (0.39) MAPTTSHRHSD17B10PARP1SMYD3
SCHEMBL7711411 0.84 PARP1 (0.40) MAPTPARP1SMYD3PDE3BPDE3A
SCHEMBL7711071 0.82 NAMPT (0.36) NAMPTRAB9ACYP17A1CYP19A1RORC
SCHEMBL7711391 0.81 SMYD3 (0.38) TSHRPARP1SMYD3PDE3BPDE3A
SCHEMBL7711428 0.81 PARP1 (0.39) PARP1SMYD3PDE3BPDE3AKDR
SCHEMBL7711067 0.80 NAMPT (0.36) MAPTTSHRHSD17B10NAMPTRAB9A
SCHEMBL7708185 0.79 PARP1 (0.40) PARP1SMYD3PDE3BPDE3AKDR
SCHEMBL7094003 0.79 ADORA2B (0.32) CYP17A1
SCHEMBL7096395 0.74 NPC1 (0.33) MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed