SCHEMBL7708185

SCHEMBL7708185

CC1Oc2ccc(C(C)(NC(=O)OC(C)(C)C)c3cccc4ccccc34)cc2NC1=O

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.40
SMYD3 Q9H7B4 3/20 0.38
MAOB P27338 1/20 0.36
ADORA2A P29274 1/20 0.36
KDR P35968 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
SSTR4 P31391 2/20 0.33
MAPK10 P53779 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
IDO1 P14902 1/20 0.33
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7094456 0.90 SSTR4 (0.35) MEN1KMT2AATMSSTR4MAPK10
SCHEMBL7711411 0.81 PARP1 (0.40) PARP1SMYD3MAOBADORA2AKDR
SCHEMBL7705092 0.81 NPSR1 (0.36) MEN1KMT2AATMSSTR4NPSR1
SCHEMBL7711103 0.81 SMYD3 (0.39) PARP1SMYD3MAOBADORA2AKDR
SCHEMBL7705086 0.80 NPSR1 (0.35) MEN1KMT2AATMSSTR4MAPK10
SCHEMBL7711428 0.80 PARP1 (0.39) PARP1SMYD3MAOBADORA2AKDR
SCHEMBL7708173 0.79 MAPT (0.39) PARP1SMYD3MAOBADORA2AKDR
SCHEMBL7711391 0.79 SMYD3 (0.38) PARP1SMYD3MAOBADORA2AKDR
SCHEMBL8253091 0.72 PARP1 (0.58) PARP1SMYD3PDE3BPDE3ABRD4
SCHEMBL7096395 0.72 NPC1 (0.33) KMT2AMAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed