SCHEMBL7708177

SCHEMBL7708177

CC1Oc2ccc(C(c3cccnc3)N(C)C(=O)OC(C)(C)C)cc2NC1=O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PARP1 P09874 6/20 0.36
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
SMYD3 Q9H7B4 3/20 0.34
KDR P35968 1/20 0.32
HTR1A P08908 1/20 0.32
HTR7 P34969 1/20 0.32
MAOB P27338 1/20 0.31
ADORA2A P29274 1/20 0.31
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP3A5 P20815 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711038 0.90 PDE4D (0.32) MAPTTSHRHSD17B10CYP3A4CYP3A5
SCHEMBL7711106 0.89 PDE3B (0.38) PARP1PDE3BPDE3ASMYD3KDR
SCHEMBL7711412 0.84 PARP1 (0.39) HSD17B10PARP1PDE3BPDE3ASMYD3
SCHEMBL7711394 0.83 PARP1 (0.36) PARP1PDE3BPDE3ASMYD3KDR
SCHEMBL7711431 0.82 PARP1 (0.37) HSD17B10PARP1PDE3BPDE3ASMYD3
SCHEMBL7711069 0.81 CYP3A4 (0.31) CYP3A4CYP3A5
SCHEMBL7708190 0.80 PARP1 (0.38) PARP1PDE3BPDE3ASMYD3KDR
SCHEMBL7710769 0.79 KDM4D (0.35)
SCHEMBL6991325 0.77 SMYD3 (0.36) MAPTTSHRHSD17B10PARP1PDE3B
SCHEMBL6992024 0.74 PARP1 (0.44) MAPTTSHRHSD17B10PARP1PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed