SCHEMBL7708190

SCHEMBL7708190

CC1Oc2ccc(C(c3cccc4ccccc34)N(C)C(=O)OC(C)(C)C)cc2NC1=O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.38
SMYD3 Q9H7B4 3/20 0.35
PDE3B Q13370 2/20 0.35
PDE3A Q14432 2/20 0.35
MAOB P27338 1/20 0.34
ADORA2A P29274 1/20 0.34
KDR P35968 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
HTR1A P08908 1/20 0.33
HTR7 P34969 1/20 0.33
BRD4 O60885 2/20 0.32
CREBBP Q92793 2/20 0.32
EDNRA P25101 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711384 0.91 EDNRA (0.31) MEN1KMT2AATMEDNRA
SCHEMBL7711412 0.83 PARP1 (0.39) PARP1SMYD3PDE3BPDE3AKDR
SCHEMBL7711431 0.81 PARP1 (0.37) PARP1SMYD3PDE3BPDE3AKDR
SCHEMBL7711106 0.81 PDE3B (0.38) PARP1SMYD3PDE3BPDE3AKDR
SCHEMBL7705087 0.81 EDNRA (0.31) MEN1KMT2AATMEDNRA
SCHEMBL7711394 0.80 PARP1 (0.36) PARP1SMYD3PDE3BPDE3AKDR
SCHEMBL7708177 0.80 MAPT (0.36) PARP1SMYD3PDE3BPDE3AMAOB
SCHEMBL6998315 0.77 SMYD3 (0.37) PARP1SMYD3PDE3BPDE3AMAOB
SCHEMBL6998103 0.75 PARP1 (0.46) PARP1SMYD3PDE3BPDE3AMAOB
SCHEMBL7713347 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed