SCHEMBL7705092

SCHEMBL7705092

CC1Oc2ccc(C(C)(NC(=O)OC(C)(C)C)c3cccc4ccccc34)cc2N=C1N

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ATM Q13315 1/20 0.33
SSTR4 P31391 2/20 0.33
NPC1 O15118 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32
NQO2 P16083 1/20 0.31
MAPK14 Q16539 1/20 0.31
KDM4A O75164 1/20 0.31
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708015 0.82 AAK1 (0.32)
SCHEMBL7708185 0.81 PARP1 (0.40) NPSR1MEN1KMT2AATMSSTR4
SCHEMBL7711556 0.81 NPC1 (0.33) KMT2ANPC1RAB9A
SCHEMBL7711071 0.80 NAMPT (0.36) RAB9A
SCHEMBL7708340 0.80 ALDH1A1 (0.32)
SCHEMBL7705086 0.76 NPSR1 (0.35) NPSR1MEN1KMT2AATMSSTR4
SCHEMBL6310050 0.69 CA1 (0.34) MEN1KMT2AGAA
SCHEMBL7704833 0.68 KDM4E (0.37) NPSR1CTSSCTSK
SCHEMBL4262988 0.66 MEN1 (0.43) MEN1KMT2AATMSSTR4NPC1
SCHEMBL7711362 0.66 PTPRB (0.40) NPSR1MEN1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed