SCHEMBL6309909

SCHEMBL6309909

CC1Oc2ccc(CN(Cc3cccc(CN(Cc4ccc(Cl)cc4Cl)C(=O)OC(C)(C)C)c3)C(=O)OC(C)(C)C)cc2NC1=S

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.33
PARP1 P09874 3/20 0.33
TP53 P04637 3/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
SLC6A3 Q01959 1/20 0.32
ALDH1A1 P00352 3/20 0.32
TSHR P16473 1/20 0.32
ALOX15 P16050 1/20 0.31
ERCC1 P07992 1/20 0.31
ERCC4 Q92889 1/20 0.31
MAPT P10636 2/20 0.31
IDO1 P14902 1/20 0.31
GLA P06280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704916 0.97 HSD17B10 (0.35) HSD17B10PARP1TP53SLC6A2SLC6A4
SCHEMBL6428132 0.92 RIPK1 (0.36) HSD17B10PARP1SMN1; SMN2HDAC3HDAC1
SCHEMBL6302996 0.91 PARP1 (0.43) HSD17B10PARP1TP53POLBSMN1; SMN2
SCHEMBL7708255 0.91 RIPK1 (0.36) HSD17B10PARP1SMN1; SMN2HDAC3HDAC1
SCHEMBL7711006 0.90 PARP1 (0.36) HSD17B10PARP1TP53POLBSMN1; SMN2
SCHEMBL6302929 0.89 PARP1 (0.35) HSD17B10PARP1HDAC3HDAC1HDAC2
SCHEMBL7708215 0.88 PARP1 (0.42) HSD17B10PARP1TP53SLC6A2SLC6A4
SCHEMBL6309617 0.87 HDAC1 (0.43) HSD17B10PARP1SMN1; SMN2HDAC3HDAC1
SCHEMBL6310115 0.87 PARP1 (0.37) HSD17B10PARP1TP53POLBSMN1; SMN2
SCHEMBL7704966 0.86 TP53 (0.37) HSD17B10PARP1TP53POLBHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6841550-B1 Benzoxazine and benzothiazine derivatives and their use in medicines SCHERING AKTIENGESELLSCHAFT (DE) 2005-01-11 US disclosed