SCHEMBL7708427

SCHEMBL7708427

Cc1ccccc1-c1cc(N)n2nc(-c3ccc(Br)o3)nc2c1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.53
NPC1 O15118 1/20 0.49
CASP3 P42574 1/20 0.49
RAB9A P51151 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
ADORA3 P0DMS8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711726 0.89 ADORA2A (0.54) ADORA2ANPC1RAB9AADORA3
SCHEMBL7705607 0.86 NPC1 (0.52) ADORA2ANPC1RAB9A
SCHEMBL7705869 0.83 ADORA2A (0.56) ADORA2ANPC1RAB9A
SCHEMBL7703126 0.82 ADORA2A (0.53) ADORA2ANPC1RAB9AADORA3
SCHEMBL7705879 0.82 ADORA2A (0.56) ADORA2A
SCHEMBL7703027 0.82 ADORA2A (0.51) ADORA2ANPC1RAB9AADORA3
SCHEMBL7708821 0.78 ADORA2A (0.54) ADORA2AADORA3
SCHEMBL7711821 0.78 ADORA2A (0.54) ADORA2AADORA3
SCHEMBL7490670 0.78 ADORA2A (0.62) ADORA2AADORA3
SCHEMBL7702974 0.78 ADORA2A (0.49) ADORA2ANPC1RAB9AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed