SCHEMBL7702974

SCHEMBL7702974

COc1ccc(-c2cc(N)n3nc(-c4ccc(Br)o4)nc3c2)c(OC)n1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.49
ADORA3 P0DMS8 1/20 0.37
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705607 0.82 NPC1 (0.52) ADORA2AKDM4EHSD17B10NPC1ALDH1A1
SCHEMBL7708987 0.78 ADORA2A (0.48) ADORA2AADORA3KDM4EHSD17B10NPC1
SCHEMBL7708427 0.78 ADORA2A (0.53) ADORA2AADORA3NPC1RAB9A
SCHEMBL7703022 0.78 NPC1 (0.56) ADORA2ANPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL7490670 0.77 ADORA2A (0.62) ADORA2AADORA3
SCHEMBL7705869 0.76 ADORA2A (0.56) ADORA2AKDM4ENPC1ALDH1A1RAB9A
SCHEMBL7703027 0.76 ADORA2A (0.51) ADORA2AADORA3KDM4ENPC1ALDH1A1
SCHEMBL7711821 0.74 ADORA2A (0.54) ADORA2AADORA3KDM4EALDH1A1SMN1; SMN2
SCHEMBL7708821 0.74 ADORA2A (0.54) ADORA2AADORA3KDM4E
SCHEMBL7703126 0.74 ADORA2A (0.53) ADORA2AADORA3NPC1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed