SCHEMBL7708511

SCHEMBL7708511

C[C@H](N)C(=O)N1CCC[C@]1(C(=O)O)C1(C)CCCCC1.N=C(N)c1ccc(C(N)=O)cn1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.32
F2 P00734 1/20 0.31
NNMT P40261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6484830 0.82 NNMT (0.32) BACE1NNMT
SCHEMBL6475187 0.81 F2 (0.33) F2
SCHEMBL6487072 0.79 DPP4 (0.36)
SCHEMBL6475867 0.70 ITGB3 (0.34)
SCHEMBL8725900 0.70 F2 (0.31) F2
SCHEMBL6486871 0.70 F2 (0.41) F2
Acetic Acid SCHEMBL6476505 0.68 NNMT (0.50) NNMT
SCHEMBL6476554 0.67 NNMT (0.57) NNMT
SCHEMBL6476401 0.67 ITGB3 (0.36) F2
SCHEMBL8807564 0.67 ITGB3 (0.33) BACE1NNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6444817-B1 ANTICOAGULANTS ABBOTT LABORATORIES 2002-09-03 US disclosed
US-6030972-A 2- OR 5-AMINOMETHYL,2- OR 5-CYANOPYRIMIDINES AS INTERMEDIATES OF ANTICOAGULANTS IN EXTRACORPOREAL CIRCULATION (HEART-LUNG MACHINE, HEMODIALYSIS) BASF AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
EP-0873356-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-10-28 EP disclosed
WO-1996025426-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1996-08-22 WO disclosed