SCHEMBL7708517

SCHEMBL7708517

COCCOc1cc2ncnc(Nc3ccc(OC)cc3)c2cc1OCCOC

nearest known ligand 0.77

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.77
LCK P06239 2/20 0.77
KDM1A O60341 1/20 0.75
KDR P35968 5/20 0.73
GAK O14976 1/20 0.71
FGFR1 P11362 1/20 0.66
FLT1 P17948 1/20 0.66
FBP1 P09467 1/20 0.66
ILK Q13418 1/20 0.65
MAPT P10636 1/20 0.64
GRM1 Q13255 1/20 0.64
HDAC3 O15379 1/20 0.64
HDAC1 Q13547 1/20 0.64
HDAC6 Q9UBN7 1/20 0.64
SRC P12931 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708102 0.92 EGFR (0.67) EGFRLCKKDM1AKDRGAK
SCHEMBL18447218 0.89 KDM1A (0.77) EGFRLCKKDM1AKDRGAK
SCHEMBL16660323 0.88 EGFR (0.77) EGFRLCKKDM1AKDRGAK
SCHEMBL28105746 0.88 KDR (0.75) EGFRKDM1AKDRGAKFGFR1
SCHEMBL20805304 0.88 EGFR (0.77) EGFRLCKKDM1AKDRGAK
SCHEMBL5472599 0.87 EGFR (1.00) EGFRLCKKDRGAKFLT1
Hydrochloric Acid SCHEMBL5479915 0.86 EGFR (1.00) EGFRLCKKDRGAKFLT1
SCHEMBL22381430 0.86 KDM1A (0.72) EGFRLCKKDM1AKDRGAK
SCHEMBL13219733 0.85 EGFR (0.78) EGFRLCKKDM1AKDRGAK
SCHEMBL30016831 0.81 EGFR (0.60) EGFRLCKKDM1AKDRGAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105884653-A Erlotinib derivative and preparing method thereof 浙江汇能生物股份有限公司 2016-08-24 CN disclosed
US-6476040-B1 Processes and intermediates for preparing anti-cancer compounds PFIZER INC. 2002-11-05 US disclosed
EP-1044969-A2 Processes and intermediates for preparing anti-cancer compounds Pfizer Products Inc. (US) 2000-10-18 EP disclosed