SCHEMBL7708776

SCHEMBL7708776

Nc1cc(-c2ccccc2Cl)cc2nc(-c3ccccn3)nn12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.53
GRM5 P41594 4/20 0.47
MAPK14 Q16539 2/20 0.46
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.40
DCTPP1 Q9H773 1/20 0.40
ADORA1 P30542 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
CHRNA7 P36544 1/20 0.38
ALOX15 P16050 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
BACE1 P56817 1/20 0.38
HPGD P15428 1/20 0.38
NFKB1 P19838 1/20 0.38
HTT P42858 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7428533 0.86 ADORA2A (0.60) ADORA2AALDH1A1SMN1; SMN2KDM4EMAPT
SCHEMBL7708534 0.86 ADORA2A (0.53) ADORA2AGRM5ALDH1A1KDM4EDCTPP1
SCHEMBL7711376 0.86 ADORA2A (0.53) ADORA2AGRM5MAPK14ALDH1A1SMN1; SMN2
SCHEMBL7708907 0.85 ADORA2A (0.52) ADORA2AGRM5ALDH1A1SMN1; SMN2KDM4E
SCHEMBL7705856 0.84 ADORA2A (0.54) ADORA2AGRM5ALDH1A1SMN1; SMN2KDM4E
SCHEMBL7428299 0.83 ADORA2A (0.53) ADORA2AGRM5ALDH1A1SMN1; SMN2KDM4E
SCHEMBL7709217 0.83 GRM5 (0.50) ADORA2AGRM5ALDH1A1SMN1; SMN2KDM4E
SCHEMBL7703127 0.82 ADORA2A (0.52) ADORA2AGRM5ALDH1A1SMN1; SMN2MAPT
SCHEMBL7705845 0.82 ADORA2A (0.49) ADORA2AGRM5SMN1; SMN2MAPTADORA1
SCHEMBL7431418 0.81 ADORA2A (0.56) ADORA2AGRM5ALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed