SCHEMBL7708534

SCHEMBL7708534

Nc1cc(-c2ccccc2F)cc2nc(-c3ccccn3)nn12

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.53
GRM5 P41594 8/20 0.49
DCTPP1 Q9H773 1/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
F2 P00734 1/20 0.40
F12 P00748 1/20 0.40
ADORA1 P30542 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALOX15 P16050 1/20 0.38
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7428533 0.86 ADORA2A (0.60) ADORA2AL3MBTL1NPC1ALDH1A1HTT
SCHEMBL7708776 0.86 ADORA2A (0.53) ADORA2AGRM5DCTPP1L3MBTL1NPC1
SCHEMBL7711376 0.86 ADORA2A (0.53) ADORA2AGRM5DCTPP1L3MBTL1NPC1
SCHEMBL7427435 0.84 ADORA2A (0.54) ADORA2AGRM5DCTPP1L3MBTL1NPC1
SCHEMBL7709217 0.83 GRM5 (0.50) ADORA2AGRM5DCTPP1NPC1ALDH1A1
SCHEMBL7708837 0.82 GRM5 (0.52) ADORA2AGRM5DCTPP1L3MBTL1NPC1
SCHEMBL7705845 0.82 ADORA2A (0.49) ADORA2AGRM5L3MBTL1NPC1HTT
SCHEMBL7431418 0.81 ADORA2A (0.56) ADORA2AGRM5L3MBTL1NPC1ALDH1A1
SCHEMBL7487093 0.81 ADORA2A (0.45) ADORA2AGRM5L3MBTL1NPC1ALDH1A1
SCHEMBL7708387 0.80 BACE1 (0.40) ADORA2AL3MBTL1NPC1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed