SCHEMBL7708869

SCHEMBL7708869

COc1ccc(-c2cc(N)n3nc(-c4ccc(C)o4)nc3c2)c(OC)c1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.49
TSHR P16473 2/20 0.43
HSD17B10 Q99714 2/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
PKM P14618 1/20 0.42
RAB9A P51151 1/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42
MAPT P10636 1/20 0.42
TLR9 Q9NR96 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
ADORA3 P0DMS8 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708420 0.88 ADORA2A (0.51) ADORA2AKDM4EALDH1A1ADORA3ADORA1
SCHEMBL7709161 0.86 ADORA2A (0.53) ADORA2AHSD17B10KDM4EALDH1A1HPGD
SCHEMBL7709024 0.84 NPC1 (0.41) ADORA2ATSHRHSD17B10KDM4EALDH1A1
SCHEMBL7709129 0.84 ADORA2A (0.56) ADORA2A
SCHEMBL7487041 0.83 ADORA2A (0.51) ADORA2AKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL7492811 0.82 ADORA2A (0.52) ADORA2ATSHRHSD17B10KDM4EALDH1A1
SCHEMBL7711726 0.78 ADORA2A (0.54) ADORA2AALDH1A1HPGDSMN1; SMN2NPC1
SCHEMBL7703002 0.78 ADORA2A (0.47) ADORA2ATSHRHSD17B10KDM4EALDH1A1
SCHEMBL7711750 0.77 ADORA2A (0.57) ADORA2AKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL7711685 0.77 ADORA2A (0.57) ADORA2AHSD17B10KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed