SCHEMBL7708420

SCHEMBL7708420

COc1ccccc1-c1cc(N)n2nc(-c3ccc(C)o3)nc2c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.51
ADORA3 P0DMS8 2/20 0.45
ADORA1 P30542 2/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705607 0.88 NPC1 (0.52) ADORA2AKDM4EALDH1A1
SCHEMBL7708869 0.88 ADORA2A (0.49) ADORA2AADORA3ADORA1KDM4EALDH1A1
SCHEMBL7711726 0.87 ADORA2A (0.54) ADORA2AADORA3ADORA1ALDH1A1
SCHEMBL7709007 0.85 ADORA2A (0.53) ADORA2AADORA3ADORA1ALDH1A1
SCHEMBL7703196 0.85 ADORA2A (0.53) ADORA2AADORA3ADORA1KDM4EALDH1A1
SCHEMBL7492811 0.84 ADORA2A (0.52) ADORA2AADORA3KDM4EALDH1A1
SCHEMBL7708829 0.84 ADORA2A (0.70) ADORA2A
SCHEMBL7711685 0.83 ADORA2A (0.57) ADORA2AADORA3ADORA1KDM4EALDH1A1
SCHEMBL7709161 0.81 ADORA2A (0.53) ADORA2AADORA3ADORA1KDM4EALDH1A1
SCHEMBL7487041 0.81 ADORA2A (0.51) ADORA2AADORA3ADORA1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed