SCHEMBL7708933

SCHEMBL7708933

Nc1cc(-c2ccc(OC(F)(F)F)cc2)cc(N)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.46
TPX2 Q9ULW0 1/20 0.46
SCN5A Q14524 8/20 0.45
SCN9A Q15858 6/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
GMNN O75496 1/20 0.45
USP2 O75604 1/20 0.45
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
GAA P10253 1/20 0.45
CYP2C9 P11712 1/20 0.45
PKM P14618 1/20 0.45
ALOX15 P16050 1/20 0.45
NFKB1 P19838 1/20 0.45
SLC6A2 P23975 1/20 0.45
SCN4A P35499 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1242144 0.78 KIF11 (0.52) AURKATPX2SCN5ASCN9ATP53
SCHEMBL3997703 0.78 AKR1C2 (0.50) AURKATPX2SCN5ASCN2AMAPK1
SCHEMBL27960724 0.77 BACE1 (0.59) SCN5ASCN9ANPC1RAB9AGMNN
SCHEMBL18654126 0.76 LTA4H (0.56) SCN5ASCN9ASCN2AALOX5APFEN1
Hydrochloric Acid SCHEMBL29386875 0.76 KIF11 (0.50) AURKATPX2SCN5ASCN9ANPC1
SCHEMBL24024734 0.76 MEN1 (0.54) AURKATPX2SCN5AGAASCN2A
SCHEMBL28563593 0.75 HDAC3 (0.49) SCN5ASCN9ANPC1RAB9AGMNN
SCHEMBL30386990 0.75 HDAC3 (0.49) SCN5ASCN9ANPC1RAB9AGMNN
SCHEMBL7708814 0.75 DYRK1A (0.65) NPC1RAB9ATP53NFKB1SMN1; SMN2
SCHEMBL7703168 0.75 KIF11 (0.59) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed