SCHEMBL7709344

SCHEMBL7709344

N#Cc1ccc(Cn2cncc2CCC(=O)O)cc1F.[LiH]

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 12/20 0.51
CYP11B2 P19099 12/20 0.51
FFAR1 O14842 2/20 0.42
FFAR4 Q5NUL3 2/20 0.42
CACNA1H O95180 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7971164 0.99 CYP11B1 (0.52) CYP11B1CYP11B2FFAR1FFAR4CACNA1H
SCHEMBL7704754 0.89 CYP11B1 (0.45) CYP11B1CYP11B2CACNA1H
Lithium Ion SCHEMBL7709340 0.88 CYP11B2 (0.50) CYP11B1CYP11B2CACNA1H
SCHEMBL6452310 0.88 CYP11B1 (0.46) CYP11B1CYP11B2CACNA1H
Bromide SCHEMBL7629321 0.87 CYP11B1 (0.45) CYP11B1CYP11B2CACNA1H
SCHEMBL7713236 0.86 CYP11B1 (0.70) CYP11B1CYP11B2CACNA1H
SCHEMBL7713277 0.83 CYP11B1 (0.46) CYP11B1CYP11B2
SCHEMBL7714120 0.83 CYP11B1 (0.52) CYP11B1CYP11B2CACNA1H
Hydrochloric Acid SCHEMBL7183805 0.83 CYP11B1 (0.47) CYP11B1CYP11B2
SCHEMBL6433915 0.83 CYP11B1 (0.64) CYP11B1CYP11B2CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441017-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2002-08-27 US disclosed
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed