SCHEMBL7704754

SCHEMBL7704754

N#Cc1ccc(Cn2cncc2CC(=O)O)cc1F.[LiH]

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 6/20 0.45
CYP11B2 P19099 6/20 0.45
CACNA1H O95180 10/20 0.43
FNTA P49354 2/20 0.42
FNTB P49356 2/20 0.42
PGGT1B P53609 2/20 0.42
CACNA1G O43497 1/20 0.41
CACNA1I Q9P0X4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6452310 0.99 CYP11B1 (0.46) CYP11B1CYP11B2CACNA1HFNTAFNTB
Bromide SCHEMBL7629321 0.98 CYP11B1 (0.45) CYP11B1CYP11B2CACNA1HFNTAFNTB
SCHEMBL7709344 0.89 CYP11B1 (0.51) CYP11B1CYP11B2CACNA1H
Lithium Ion SCHEMBL7704749 0.88 CYP11B2 (0.44) CYP11B1CYP11B2CACNA1HFNTAFNTB
SCHEMBL7971164 0.88 CYP11B1 (0.52) CYP11B1CYP11B2CACNA1H
SCHEMBL7704743 0.86 CYP11B1 (0.55) CYP11B1CYP11B2CACNA1HFNTAFNTB
SCHEMBL6433915 0.84 CYP11B1 (0.64) CYP11B1CYP11B2CACNA1H
SCHEMBL6410255 0.81 CYP11B2 (0.47) CYP11B1CYP11B2CACNA1HFNTAFNTB
Hydrochloric Acid SCHEMBL2789879 0.81 CYP11B1 (0.47) CYP11B1CYP11B2CACNA1HFNTAFNTB
Lithium Ion SCHEMBL7709340 0.81 CYP11B2 (0.50) CYP11B1CYP11B2CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
US-6358985-B1 ANTICANCER AGENT MERCK & CO., INC. 2002-03-19 US disclosed
EP-1091736-A4 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 2001-10-24 EP disclosed
EP-1091736-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2001-04-18 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed
WO-2000001382-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2000-01-13 WO disclosed