SCHEMBL7709632

SCHEMBL7709632

CC(C)(C)ON1C(=O)c2cccc3c(Br)ccc(c23)C1=O

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 16/20 0.58
ALDH1A1 P00352 2/20 0.51
POLB P06746 2/20 0.51
RXFP1 Q9HBX9 1/20 0.51
LMNA P02545 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
NPC1 O15118 1/20 0.50
MAPT P10636 1/20 0.50
PABPC1 P11940 1/20 0.50
KMT2A Q03164 1/20 0.50
TP53 P04637 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
THRB P10828 1/20 0.48
TLR9 Q9NR96 1/20 0.48
S1PR2 O95136 1/20 0.48
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13495353 0.83 CYP1B1 (0.63) CYP1B1ALDH1A1POLBRXFP1LMNA
SCHEMBL28064300 0.79 CYP1B1 (0.67) CYP1B1ALDH1A1POLBRXFP1LMNA
SCHEMBL7712213 0.79 PRMT1 (0.46) CYP1B1ALDH1A1POLBLMNAKDM4E
SCHEMBL30905987 0.78 CYP1B1 (0.69) CYP1B1ALDH1A1POLBRXFP1LMNA
SCHEMBL4866412 0.78 CYP1B1 (0.69) CYP1B1ALDH1A1POLBRXFP1LMNA
SCHEMBL7703735 0.76 KDM4E (0.44) ALDH1A1POLBLMNAKDM4EMEN1
SCHEMBL7850554 0.75 GAA (0.47) ALDH1A1LMNAKDM4EMEN1MAPT
SCHEMBL7703829 0.74 POLB (0.65) CYP1B1ALDH1A1POLBRXFP1LMNA
SCHEMBL29074524 0.74 CYP1B1 (0.64) CYP1B1ALDH1A1POLBRXFP1LMNA
SCHEMBL17792909 0.74 CYP1B1 (0.63) CYP1B1ALDH1A1POLBRXFP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed