SCHEMBL7709738

SCHEMBL7709738

COc1cc2c(cc1O)NC(=O)[C@H]1C[C@@H](O)CN1C2=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.41
ACHE P22303 2/20 0.38
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 4/20 0.33
CHEK1 O14757 2/20 0.33
PTGS2 P35354 1/20 0.32
MAPT P10636 3/20 0.32
HPGD P15428 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
PARP1 P09874 1/20 0.32
CGAS Q8N884 1/20 0.32
GAA P10253 1/20 0.32
CDC7 O00311 1/20 0.32
DAPK3 O43293 1/20 0.32
DYRK3 O43781 1/20 0.32
MAP4K4 O95819 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10771699 1.00 EGFR (0.41) EGFRACHEHTR2AHTR2CHTR2B
SCHEMBL12856769 0.92 KDM4E (0.38) HTR2AHTR2CHTR2BKDM4EALDH1A1
SCHEMBL13422023 0.84 KDM4E (0.37) HTR2AHTR2CHTR2BKDM4EALDH1A1
SCHEMBL5926038 0.84 KDM4E (0.37) HTR2AHTR2CHTR2BKDM4EALDH1A1
SCHEMBL16067443 0.83 POLB (0.40) HTR2AHTR2CHTR2BKDM4EMAPT
SCHEMBL7709742 0.83 EGFR (0.37) EGFRACHEHTR2AHTR2CHTR2B
SCHEMBL23837196 0.80 EGFR (0.35) EGFRACHEHTR2AHTR2CHTR2B
SCHEMBL12347418 0.80 KDM4E (0.35) HTR2AHTR2CHTR2BKDM4EALDH1A1
SCHEMBL29778202 0.80 PDE3B (0.44) HTR2AHTR2CHTR2BKDM4EALDH1A1
SCHEMBL20863884 0.80 ALOX15 (0.47) EGFRACHEHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362331-B1 PYRROLO(2,1-C)(1,4)BENZODIAZEPINE COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2002-03-26 US disclosed