SCHEMBL7710679

SCHEMBL7710679

CCCN(CCC)c1c(N[C@@H](Cc2ccc(Nc3nc(CC)cc4cc(OC)ccc34)cc2)C(=O)OCC)c(=O)c1=O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 10/20 0.42
ITGA4 P13612 10/20 0.42
TP53 P04637 1/20 0.35
PTGDR Q13258 1/20 0.33
CRHR1 P34998 2/20 0.33
ELANE P08246 1/20 0.33
SLC2A1 P11166 1/20 0.33
ALDH1A1 P00352 1/20 0.32
KDR P35968 1/20 0.32
MAPT P10636 1/20 0.32
KDM1A O60341 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7714172 0.94 ITGB1 (0.49) ITGB1ITGA4TP53PTGDRELANE
SCHEMBL7714181 0.93 ITGB1 (0.51) ITGB1ITGA4PTGDR
SCHEMBL7714205 0.86 ITGB1 (0.58) ITGB1ITGA4PTGDRKDM1A
SCHEMBL7716171 0.85 TP53 (0.36) ITGB1ITGA4TP53PTGDRELANE
SCHEMBL7716181 0.85 TP53 (0.36) ITGB1ITGA4TP53PTGDRELANE
SCHEMBL7715527 0.83 TP53 (0.34) ITGB1ITGA4TP53PTGDRELANE
SCHEMBL7715520 0.83 TP53 (0.34) ITGB1ITGA4TP53PTGDRELANE
SCHEMBL7714179 0.81 ITGB1 (0.49) ITGB1ITGA4
SCHEMBL7715542 0.79 ITGB1 (0.41) ITGB1ITGA4TP53ELANEALDH1A1
SCHEMBL7716449 0.75 ITGB1 (0.41) ITGB1ITGA4PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403608-B1 ANTIINFLAMMATORY AND IMMUNE DISORDERS CELLTECH R&D, LTD. (GB) 2002-06-11 US disclosed