SCHEMBL7712413

SCHEMBL7712413

CS(=O)(=O)N1CCN(c2nc(N)ncc2Oc2ccc(Cl)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.46
BCR P11274 1/20 0.46
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
DHFR P00374 1/20 0.39
MTOR P42345 4/20 0.39
PIK3CD O00329 3/20 0.39
PIK3R1 P27986 3/20 0.39
PIK3CA P42336 3/20 0.39
PIK3CB P42338 3/20 0.39
PIK3CG P48736 3/20 0.39
HRH4 Q9H3N8 2/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7714275 0.85 POLB (0.48) ABL1BCRNPSR1HTTSMN1; SMN2
SCHEMBL7708416 0.85 HRH4 (0.55) DHFRHRH4
SCHEMBL7708563 0.82 PI4KB (0.46) DHFRALDH1A1PI4KB
SCHEMBL7708471 0.82 DHFR (0.41) HTTSMN1; SMN2DHFRHRH4PI4KB
SCHEMBL7714398 0.82 KDM4E (0.43) NPC1RAB9AHTTDHFRHRH4
SCHEMBL7712369 0.81 DHFR (0.50) CNR1NPC1RAB9ANPSR1HTT
SCHEMBL7714137 0.80 LTA4H (0.51) DHFRHRH4
SCHEMBL7714247 0.80 MEN1 (0.53) NPSR1HTTDHFRMTORPIK3R1
SCHEMBL7714733 0.79 PDGFRB (0.43) MAPK1PI4KB
SCHEMBL7714261 0.79 MAPT (0.50) RAB9ANPSR1SMN1; SMN2ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6440965-B1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system KRENITSKY PHARMACEUTICALS, INC. 2002-08-27 US claimed
US-6440965-B1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system KRENITSKY PHARMACEUTICALS, INC. 2002-08-27 US disclosed