SCHEMBL7713258

SCHEMBL7713258

CN[C@H]1CCSC2c3ccccc3CC(C)N2C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
SLC6A4 P31645 1/20 0.40
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40
HTR2B P41595 1/20 0.40
KCNH2 Q12809 1/20 0.40
PDPK1 O15530 1/20 0.39
PRCP P42785 1/20 0.36
ACE P12821 3/20 0.34
MME P08473 2/20 0.34
XIAP P98170 4/20 0.33
BIRC3 Q13489 4/20 0.33
BIRC2 Q13490 4/20 0.33
SIGMAR1 Q99720 1/20 0.32
OPRM1 P35372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14170111 0.73 BRD4 (0.38) ADRA2AADRA2BADRA2CSLC6A2HTR2A
SCHEMBL12747426 0.73 ACE (0.50) ADRA2AADRA2BADRA2CSLC6A2HTR2A
SCHEMBL14170247 0.71 XIAP (0.38) ADRA2AADRA2BADRA2CSLC6A2HTR2A
SCHEMBL14169932 0.71 ADRA2A (0.43) ADRA2AADRA2BADRA2CSLC6A2HTR2A
SCHEMBL14169897 0.70 OPRM1 (0.40) PDPK1PRCPXIAPBIRC3BIRC2
SCHEMBL14170126 0.69 ADRA2A (0.42) ADRA2AADRA2BADRA2CSLC6A2HTR2A
SCHEMBL12747479 0.68 ACE (0.40) ADRA2AADRA2BADRA2CSLC6A2HTR2A
SCHEMBL14392106 0.67 PRCP (0.38) HTR2AHTR2CHTR2BPRCPOPRM1
SCHEMBL10060256 0.67 PRCP (0.38) HTR2AHTR2CHTR2BPRCPOPRM1
SCHEMBL14170136 0.66 ADRA2A (0.50) ADRA2AADRA2BADRA2CSLC6A2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6509330-B2 Angiotensin converting enzyme (ACE); neutral endopeptidase (NEP); containing a dipeptide derived from an amino acid, or a conformationally restricted dipeptide mimic BRISTOL-MYERS SQUIBB COMPANY 2003-01-21 US disclosed