SCHEMBL7714152

SCHEMBL7714152

CN1CCN(c2nc(Cl)ncc2Oc2ccc(Cl)cc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 12/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
NPC1 O15118 1/20 0.42
GAA P10253 1/20 0.42
RAB9A P51151 1/20 0.42
HTR3A P46098 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA1 P30542 1/20 0.41
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708416 0.87 HRH4 (0.55) HRH4HTR1ADRD2
SCHEMBL7716722 0.85 HRH4 (0.51) HRH4NPC1GAARAB9AHTR3A
SCHEMBL7714260 0.85 HRH4 (0.51) HRH4SMN1; SMN2NPC1GAARAB9A
SCHEMBL7714501 0.84 LMNA (0.46) HRH4SMN1; SMN2GAARAB9AHTR1A
SCHEMBL7714712 0.82 KMT2A (0.54) HRH4HTR3A
SCHEMBL7708460 0.82 KMT2A (0.54) HRH4HTR3A
SCHEMBL7716613 0.82 HRH4 (0.52) HRH4SMN1; SMN2NPC1GAARAB9A
SCHEMBL7714490 0.81 ALK (0.53) HRH4
SCHEMBL7716737 0.80 ALDH1A1 (0.48) HRH4SMN1; SMN2GAARAB9AHTR3A
SCHEMBL7714132 0.79 HRH4 (0.53) HRH4HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6440965-B1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system KRENITSKY PHARMACEUTICALS, INC. 2002-08-27 US disclosed