SCHEMBL7714348

SCHEMBL7714348

COc1ccc(-c2ncnc3cc(OC)c(OC)cc23)c(F)c1

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KIT P10721 11/20 0.74
EGFR P00533 6/20 0.54
KDR P35968 2/20 0.54
LCK P06239 2/20 0.50
TRPA1 O75762 1/20 0.49
PDE10A Q9Y233 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15504611 0.85 KIT (1.00) KITEGFRKDRTRPA1
SCHEMBL15665140 0.78 KIT (1.00) KIT
SCHEMBL2926080 0.76 KIT (0.67) KITEGFRKDRTRPA1PDE10A
SCHEMBL1264612 0.76 KIT (0.60) KITEGFRKDRLCKTRPA1
SCHEMBL6182448 0.75 KIT (0.78) KITEGFRKDRTRPA1
SCHEMBL15664429 0.74 KIT (1.00) KIT
SCHEMBL15664700 0.74 KIT (1.00) KIT
SCHEMBL17780990 0.74 AMY1A (0.52) KITEGFRTRPA1
SCHEMBL15665218 0.73 KIT (1.00) KIT
SCHEMBL6836832 0.72 EGFR (0.62) KITEGFRKDRLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37650-E1 Aryl and heteroaryl quinazoline compounds which inhibit CSF-1R receptor tyrosine kinase AVENTIS PHARMACETICAL PRODUCTS, INC. 2002-04-09 US claimed