SCHEMBL7715181

SCHEMBL7715181

C=CCC(C(=O)O)(C(=O)O)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.67
TSHR P16473 1/20 0.67
HTT P42858 1/20 0.58
KMT2A Q03164 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
MEN1 O00255 1/20 0.45
CYP1A2 P05177 3/20 0.42
CYP2C19 P33261 4/20 0.39
MAPT P10636 2/20 0.39
HIF1A Q16665 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP3A4 P08684 2/20 0.38
AKT1 P31749 1/20 0.38
ATM Q13315 1/20 0.36
CYP2D6 P10635 1/20 0.36
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
AKR1B1 P15121 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7490885 0.82 ALDH1A1 (0.51) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL3593284 0.80 KCNN4 (0.53) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL7769347 0.80 ALDH1A1 (1.00) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL8358191 0.80 ALDH1A1 (0.67) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL6944126 0.80 ALDH1A1 (0.67) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL7385780 0.80 ALDH1A1 (0.67) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL5325708 0.80 ALDH1A1 (0.67) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL29220422 0.79 ALDH1A1 (0.51) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL1908316 0.78 ALDH1A1 (0.65) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL3613086 0.78 ALDH1A1 (0.65) ALDH1A1TSHRHTTKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781778-B1 Paclitaxel prodrugs, method for preparation as well as their use in selective chemotherapy PHARMACHEMIE BV (NL) 2002-04-17 EP disclosed
US-5760072-A ANTITUMOR AGENTS PHARMACHEMIE B.V. (NL) 1998-06-02 US disclosed
EP-0781778-A1 Novel paclitaxel prodrugs, method for preparation as well as their use in selective chemotherapy PHARMACHEMIE B.V. (NL) 1997-07-02 EP disclosed