SCHEMBL7715307

SCHEMBL7715307

COC(=O)c1ccc(C#CC(O)c2ccc3c(c2)OCCC3(SC)SC)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 3/20 0.38
RARG P13631 3/20 0.38
RARA P10276 2/20 0.38
KDM4E B2RXH2 6/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
TSHR P16473 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ACACB O00763 1/20 0.34
CYP3A4 P08684 4/20 0.33
PTPN11 Q06124 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
TP53 P04637 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7715091 0.93 RARB (0.42) RARBRARGRARAKDM4EALDH1A1
SCHEMBL7709290 0.89 RARB (0.41) RARBRARGRARAACACBCYP3A4
SCHEMBL7715267 0.87 CA12 (0.35) KDM4EALDH1A1ACACBPTPN11GAA
SCHEMBL7709229 0.82 RARB (0.41) RARBRARGRARAACACBCYP3A4
SCHEMBL8681441 0.81 NPC1 (0.33) RARBRARGRARANPC1RAB9A
SCHEMBL7709302 0.80 KDM4C (0.32) KDM4EALDH1A1HPGDHSD17B10CYP2C9
SCHEMBL7714840 0.80 CA12 (0.35) RARBRARGRARAKDM4EALDH1A1
SCHEMBL7713112 0.79 RARB (0.41) RARBRARGRARAACACBCYP3A4
SCHEMBL7715161 0.77 CYP3A4 (0.54) RARBRARGRARAKDM4EALDH1A1
SCHEMBL4847717 0.74 CYP3A4 (0.38) RARBRARGRARAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6368608-B1 SKIN DISORDERS CENTRE INTERNATIONAL DE RECHERCHE DERMATOLOGIQUES GALDERMA (C.I.R.D.) (FR) 2002-04-09 US disclosed
US-6162445-A Polyaromatic propynyl compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2000-12-19 US disclosed
US-5716624-A USEFUL FOR TREATING DERMATOLOGICAL, RHEUMATIC, RESPIRATORY, CARDIOVASCULAR, OPTHALMOLOGICAL DISORDERS, AS WELL AS MAMMALIAN SKIN AND HAIR CONDITIONS/DISORDERS C.I.R.D. GALDERMA (FR) 1998-02-10 US disclosed