SCHEMBL7714840

SCHEMBL7714840

COC(=O)c1ccc(C#CC(O)c2ccc3c(c2)C(SC)(SC)CCO3)cc1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK4 Q16654 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
ACACB O00763 1/20 0.34
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.30
MAPT P10636 1/20 0.30
ADRB2 P07550 1/20 0.30
ADRB1 P08588 1/20 0.30
ADRB3 P13945 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7715267 0.93 CA12 (0.35) CA12CA1CA2CA7PDK2
SCHEMBL7713267 0.90 ACACB (0.33) ACACBRARARARBRARGKDM4E
SCHEMBL8440033 0.88 CA12 (0.41) CA12CA1CA2CA7PDK2
SCHEMBL7715091 0.87 RARB (0.42) ACACBRARARARBRARGKDM4E
SCHEMBL7709302 0.83 KDM4C (0.32) ACACBKDM4EALDH1A1
SCHEMBL7714849 0.82 RARB (0.39) CA12CA1CA2CA7PDK2
SCHEMBL7709229 0.81 RARB (0.41) ACACBRARARARBRARG
SCHEMBL7715307 0.80 RARB (0.38) ACACBRARARARBRARGKDM4E
SCHEMBL7713112 0.80 RARB (0.41) ACACBRARARARBRARG
SCHEMBL8907353 0.79 CYP3A4 (0.40) CA12CA1CA2CA7PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6162445-A Polyaromatic propynyl compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2000-12-19 US claimed
EP-0661258-B1 Biaromatic propynyl compounds, pharmaceutical compositions and cosmetics containing them and their uses CIRD GALDERMA (FR) 1998-04-08 EP claimed
US-6368608-B1 SKIN DISORDERS CENTRE INTERNATIONAL DE RECHERCHE DERMATOLOGIQUES GALDERMA (C.I.R.D.) (FR) 2002-04-09 US disclosed
US-6162445-A Polyaromatic propynyl compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2000-12-19 US disclosed