SCHEMBL7715525

SCHEMBL7715525

CCc1cc2cc(OC)ccc2c(Nc2ccc(C(CC)C(Nc3c(N4C(C)CCC4C)c(=O)c3=O)C(=O)O)cc2)n1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.33
AKR1C2 P52895 3/20 0.33
AKR1C1 Q04828 1/20 0.33
PTGS1 P23219 1/20 0.33
TP53 P04637 1/20 0.31
BTK Q06187 1/20 0.31
CYP26A1 O43174 1/20 0.30
PHLPP2 Q6ZVD8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7716444 0.85 ITGB1 (0.41)
SCHEMBL7716446 0.85 ITGB1 (0.41)
SCHEMBL7716176 0.84 AKR1C3 (0.36) AKR1C3AKR1C2AKR1C1PTGS1TP53
SCHEMBL7715520 0.81 TP53 (0.34) TP53
SCHEMBL7715530 0.81 ACP1 (0.32) TP53
SCHEMBL7710707 0.71 ITGB1 (0.39)
SCHEMBL7259930 0.71 ITGB1 (0.42)
SCHEMBL5262865 0.69 MAPT (0.33)
SCHEMBL7714172 0.65 ITGB1 (0.49) TP53
SCHEMBL7718447 0.64 ITGB1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403608-B1 ANTIINFLAMMATORY AND IMMUNE DISORDERS CELLTECH R&D, LTD. (GB) 2002-06-11 US disclosed