SCHEMBL7716176

SCHEMBL7716176

CCc1cc2cc(OC)ccc2c(Nc2ccc(C(CC)C(Nc3c(OC(C)C)c(=O)c3=O)C(=O)O)cc2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 7/20 0.36
AKR1C2 P52895 7/20 0.36
PTGS1 P23219 3/20 0.36
AKR1C1 Q04828 1/20 0.36
TP53 P04637 2/20 0.33
MAPT P10636 2/20 0.33
ATM Q13315 1/20 0.32
PTGS2 P35354 3/20 0.32
CDC42 P60953 1/20 0.32
RAC1 P63000 1/20 0.32
CYP1A2 P05177 1/20 0.32
TSHR P16473 1/20 0.32
SLC22A6 Q4U2R8 1/20 0.32
SLC2A1 P11166 1/20 0.32
PHLPP2 Q6ZVD8 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RORC P51449 1/20 0.32
CSF1R P07333 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7715525 0.84 AKR1C3 (0.33) AKR1C3AKR1C2PTGS1AKR1C1TP53
SCHEMBL7716181 0.80 TP53 (0.36) TP53MAPTSLC2A1ALDH1A1SMN1; SMN2
SCHEMBL7716185 0.80 TP53 (0.33) AKR1C3AKR1C2PTGS1AKR1C1TP53
SCHEMBL7716171 0.80 TP53 (0.36) TP53MAPTSLC2A1ALDH1A1SMN1; SMN2
SCHEMBL7105520 0.78 F7 (0.36) TP53MAPTSMN1; SMN2HDAC1
SCHEMBL7714235 0.77 MAPT (0.36) TP53MAPTCYP1A2TSHRALDH1A1
SCHEMBL7714210 0.73 ITGB1 (0.42)
SCHEMBL7714207 0.73 ITGB1 (0.42)
SCHEMBL7260147 0.71 RAB9A (0.36) TP53MAPTALDH1A1SMN1; SMN2
SCHEMBL7714205 0.71 ITGB1 (0.58) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403608-B1 ANTIINFLAMMATORY AND IMMUNE DISORDERS CELLTECH R&D, LTD. (GB) 2002-06-11 US disclosed