SCHEMBL7715904

SCHEMBL7715904

c1ccc2c(c1)CCCN2c1cc2ccccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
ALOX15 P16050 1/20 0.46
BRCA1 P38398 1/20 0.46
ROCK1 Q13464 1/20 0.45
ALDH1A1 P00352 4/20 0.44
HPGD P15428 3/20 0.44
KDM4C Q9H3R0 2/20 0.44
NUDT1 P36639 1/20 0.43
MAPT P10636 3/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
JAK2 O60674 1/20 0.41
JAK3 P52333 1/20 0.41
PTK2 Q05397 1/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4A O75164 1/20 0.39
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29713612 0.91 TSHR (0.55) TSHRALOX15BRCA1ROCK1ALDH1A1
SCHEMBL930442 0.91 TSHR (0.55) TSHRALOX15BRCA1ROCK1ALDH1A1
SCHEMBL27946461 0.82 ALDH1A1 (0.43) TSHRALOX15BRCA1ROCK1ALDH1A1
SCHEMBL9462932 0.79 AOC3 (0.41) TSHRALDH1A1HPGDMAPTKDM4E
2-Methylindole SCHEMBL28819401 0.79 NUDT1 (0.41) TSHRALOX15BRCA1ROCK1ALDH1A1
Trifluoromethanesulfonic Acid SCHEMBL21408184 0.79 TSHR (0.46) TSHRALOX15BRCA1ALDH1A1HPGD
Trifluoromethanesulfonic Acid SCHEMBL30159123 0.79 TSHR (0.46) TSHRALOX15BRCA1ALDH1A1HPGD
SCHEMBL7384299 0.78 TSHR (0.43) TSHRALOX15BRCA1ROCK1ALDH1A1
SCHEMBL28670716 0.77 AOC3 (0.39) HPGDMAPTKMT2AMEN1KDM4E
SCHEMBL16114138 0.72 ROCK1 (0.46) TSHRALOX15BRCA1ROCK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376670-B1 BACTERICIDE FOR GRAMPOSITIVE BACTERIA SEPRACOR INC. 2002-04-23 US disclosed
US-6103905-A EFFECTIVE AGAINST DRUG RESISTANT GRAMPOSITIVE BACTERIAL INFECTIONS; ANTIBIOTICS SEPRACOR, INC. (US) 2000-08-15 US disclosed
WO-2000034265-A2 QUINOLINE-INDOLE ANTIMICROBIAL AGENTS SEPRACOR, INC. (US) 2000-06-15 WO disclosed