SCHEMBL7716154

SCHEMBL7716154

CCCCCCNCc1[c]cccc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
LMNA P02545 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
CYP1A2 P05177 3/20 0.44
CYP2D6 P10635 3/20 0.44
CYP2C19 P33261 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
MAOA P21397 1/20 0.43
CHRM2 P08172 2/20 0.42
EPHX1 P07099 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HTT P42858 1/20 0.40
TSHR P16473 1/20 0.39
CA12 O43570 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8995479 0.98 HRH4 (0.47) HRH4HRH3LMNASIGMAR1CYP1A2
SCHEMBL8995217 0.93 HRH4 (0.41) HRH4HRH3LMNASIGMAR1CYP1A2
SCHEMBL7715270 0.86 MAOA (0.36) HRH4HRH3SIGMAR1MEN1KMT2A
SCHEMBL16892533 0.85 SIGMAR1 (0.51) HRH4HRH3LMNASIGMAR1CYP1A2
SCHEMBL16935742 0.79 MC4R (0.46) CYP1A2CYP2C19MEN1KMT2AMAOA
SCHEMBL9654441 0.79 MC4R (0.43) LMNASIGMAR1MEN1KMT2AMAOA
SCHEMBL2090459 0.78 GAA (0.34) CYP2D6HTTTSHR
SCHEMBL16892600 0.78 SIGMAR1 (0.46) SIGMAR1KMT2AALDH1A1HTTTSHR
SCHEMBL258262 0.77 KCNH2 (0.46) LMNACHRM2ALDH1A1
SCHEMBL3673115 0.77 KCNH2 (0.46) LMNACHRM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6391916-B1 ANTITUMOR AGENTS THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2002-05-21 US claimed
US-6391916-B1 ANTITUMOR AGENTS THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2002-05-21 US disclosed
US-5496844-A Indole derivatives OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1996-03-05 US disclosed
EP-0639567-A1 INDOLE DERIVATIVE OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1995-02-22 EP disclosed