SCHEMBL7716908

SCHEMBL7716908

CCN1CC[C@H](NS(=O)(=O)c2ccc(CNC3CCCC3)cc2)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.48
RECQL P46063 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
FABP6 P51161 1/20 0.46
ALDH1A1 P00352 4/20 0.45
LMNA P02545 2/20 0.45
GAA P10253 1/20 0.45
HRH3 Q9Y5N1 4/20 0.45
KCNH2 Q12809 2/20 0.45
CYP3A4 P08684 1/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
THRB P10828 1/20 0.44
HTR1A P08908 2/20 0.43
DRD2 P14416 2/20 0.43
HTR7 P34969 2/20 0.43
HTR6 P50406 2/20 0.43
BCHE P06276 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2555109 1.00 KDM4E (0.48) KDM4ERECQLSMN1; SMN2HRH2HRH1
SCHEMBL2547933 1.00 KDM4E (0.48) KDM4ERECQLSMN1; SMN2HRH2HRH1
Hydrochloric Acid SCHEMBL2552429 0.99 KDM4E (0.47) KDM4ERECQLSMN1; SMN2HRH2HRH1
Hydrochloric Acid SCHEMBL2552428 0.99 KDM4E (0.47) KDM4ERECQLSMN1; SMN2HRH2HRH1
SCHEMBL2555154 0.95 KDM4E (0.48) KDM4ERECQLSMN1; SMN2FABP6ALDH1A1
SCHEMBL7716923 0.93 SMN1; SMN2 (0.54) KDM4ERECQLSMN1; SMN2FABP6ALDH1A1
SCHEMBL2549964 0.90 KCNH2 (0.49) HRH2HRH1ALDH1A1LMNAHRH3
SCHEMBL2554540 0.87 KDM4E (0.47) KDM4ERECQLSMN1; SMN2FABP6ALDH1A1
SCHEMBL2577934 0.86 KCNH2 (0.46) HRH2HRH1HRH3KCNH2HTT
SCHEMBL2552379 0.83 HRH3 (0.45) KDM4ERECQLSMN1; SMN2HRH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011121309-A1 PHENYL SULFONYL DERIVATIVES AND THEIR USE AS HISTAMINE H3 ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-10-06 WO disclosed