SCHEMBL2552379

SCHEMBL2552379

CCN1CCC(NS(=O)(=O)c2ccc(CN(C)C3CCCC3)cc2)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.45
HRH4 Q9H3N8 1/20 0.44
HRH2 P25021 2/20 0.44
HRH1 P35367 2/20 0.44
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GAA P10253 2/20 0.42
HTT P42858 2/20 0.42
THRB P10828 1/20 0.42
KDM4E B2RXH2 1/20 0.42
RECQL P46063 1/20 0.42
HTR1A P08908 3/20 0.41
DRD2 P14416 3/20 0.41
HTR7 P34969 3/20 0.41
HTR6 P50406 3/20 0.41
KCNH2 Q12809 2/20 0.41
LMNA P02545 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2555109 0.83 KDM4E (0.48) HRH3HRH2HRH1ALDH1A1SMN1; SMN2
SCHEMBL2547933 0.83 KDM4E (0.48) HRH3HRH2HRH1ALDH1A1SMN1; SMN2
SCHEMBL7716908 0.83 KDM4E (0.48) HRH3HRH2HRH1ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL2552428 0.82 KDM4E (0.47) HRH3HRH2HRH1ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL2552429 0.82 KDM4E (0.47) HRH3HRH2HRH1ALDH1A1SMN1; SMN2
SCHEMBL2555154 0.79 KDM4E (0.48) HRH3ALDH1A1SMN1; SMN2GAAHTT
SCHEMBL7716923 0.78 SMN1; SMN2 (0.54) HRH3ALDH1A1SMN1; SMN2GAAHTT
Hydrochloric Acid SCHEMBL9796292 0.78 ALDH1A1 (0.55) HRH2HRH1ALDH1A1HTTTHRB
SCHEMBL2549964 0.76 KCNH2 (0.49) HRH3HRH2HRH1ALDH1A1HTT
SCHEMBL2552414 0.76 HRH3 (0.55) HRH3HRH2HRH1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011121309-A1 PHENYL SULFONYL DERIVATIVES AND THEIR USE AS HISTAMINE H3 ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-10-06 WO disclosed
WO-2011121309-A1 PHENYL SULFONYL DERIVATIVES AND THEIR USE AS HISTAMINE H3 ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-10-06 WO disclosed