SCHEMBL7719950

SCHEMBL7719950

C[C@@H](CCCC=CCCCC(=O)O)N(CC(O[SiH](C)C)C(C)(C)C)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.36
EPHX2 P34913 1/20 0.31
PPARG P37231 3/20 0.31
TOP1 P11387 2/20 0.31
ALDH1A1 P00352 2/20 0.31
CYP19A1 P11511 2/20 0.31
KMT2A Q03164 2/20 0.31
PPARD Q03181 2/20 0.31
PPARA Q07869 2/20 0.31
F7 P08709 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
F3 P13726 1/20 0.31
RXRA P19793 1/20 0.31
PTGS1 P23219 1/20 0.31
OXER1 Q8TDS5 1/20 0.31
USP2 O75604 2/20 0.30
CYP3A4 P08684 2/20 0.30
RECQL P46063 2/20 0.30
BLM P54132 2/20 0.30
HSD17B10 Q99714 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7805335 1.00 HDAC6 (0.36) HDAC6EPHX2PPARGTOP1ALDH1A1
SCHEMBL7719949 0.73 EPHX2 (0.33) HDAC6EPHX2PPARGTOP1ALDH1A1
SCHEMBL7805334 0.73 EPHX2 (0.33) HDAC6EPHX2PPARGTOP1ALDH1A1
SCHEMBL28675520 0.67 HDAC6 (0.33) HDAC6EPHX2KMT2ACYP1A2POLB
SCHEMBL5381165 0.64 TOP1 (0.58) PPARGTOP1ALDH1A1CYP19A1KMT2A
SCHEMBL5381163 0.64 TOP1 (0.58) PPARGTOP1ALDH1A1CYP19A1KMT2A
SCHEMBL567545 0.62 CA14 (0.31) HDAC6HDAC1HDAC2
SCHEMBL25124155 0.62 HDAC6 (0.33) HDAC6TDP1
SCHEMBL29076008 0.62 GABRP (0.34) HDAC6CYP1A2CYP2C9CYP2C19HDAC1
SCHEMBL29076007 0.62 GABRP (0.34) HDAC6CYP1A2CYP2C9CYP2C19HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6384026-B1 Macrocyclic polyamine lactones and derivatives thereof and their use as arthropod repellents CORNELL RESEARCH FOUNDATION, INC. 2002-05-07 US disclosed
EP-1067921-A4 MACROCYCLIC POLYAMINE LACTONES AND DERIVATIVES THEREOF AND THEIR USE AS ARTHROPOD REPELLENTS CORNELL RES FOUNDATION INC (US) 2001-06-27 EP disclosed
EP-1067921-A1 MACROCYCLIC POLYAMINE LACTONES AND DERIVATIVES THEREOF AND THEIR USE AS ARTHROPOD REPELLENTS CORNELL RESEARCH FOUNDATION (US) 2001-01-17 EP disclosed
WO-1999051222-A1 MACROCYCLIC POLYAMINE LACTONES AND DERIVATIVES THEREOF AND THEIR USE AS ARTHROPOD REPELLENTS CORNELL RESEARCH FOUNDATION, INC. (US) 1999-10-14 WO disclosed