SCHEMBL7721955

SCHEMBL7721955

CC(C)(C)OC(=O)N1C[C@@H](N(C(=O)CN)C(=O)OC(C)(C)C)C[C@@H]1COc1ccc(-c2ccccc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.40
SRC P12931 8/20 0.40
GPR119 Q8TDV5 1/20 0.39
USP30 Q70CQ3 1/20 0.39
MCL1 Q07820 3/20 0.37
NR1D1 P20393 1/20 0.37
FFAR4 Q5NUL3 1/20 0.36
MMP13 P45452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7733554 1.00 HDAC8 (0.40) HDAC8SRCGPR119USP30MCL1
SCHEMBL7722035 0.92 HDAC8 (0.39) HDAC8SRCUSP30FFAR4MMP13
SCHEMBL7733463 0.92 HDAC8 (0.39) HDAC8SRCUSP30FFAR4MMP13
SCHEMBL8150172 0.78 NR1H2 (0.39) SRC
SCHEMBL7721935 0.78 NR1H2 (0.39) SRC
SCHEMBL7722122 0.78 NR1H2 (0.39) SRC
SCHEMBL7727252 0.77 KDM4E (0.46) HDAC8MCL1
SCHEMBL7731479 0.76 HDAC8 (0.44) HDAC8
SCHEMBL7727102 0.76 USP30 (0.40) HDAC8GPR119USP30
SCHEMBL7726796 0.76 USP30 (0.40) HDAC8GPR119USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed
WO-2000001714-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed