SCHEMBL7721971

SCHEMBL7721971

CCOC(=O)C[C@H](NC(=O)CCCCc1ccc(C(=N)N)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)OCC

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.58
ITGA2B P08514 7/20 0.58
F2 P00734 4/20 0.51
F10 P00742 4/20 0.47
PRSS1 P07477 1/20 0.47
CTSG P08311 1/20 0.46
CMA1 P23946 1/20 0.46
ALDH1A1 P00352 1/20 0.44
HDAC1 Q13547 3/20 0.43
HDAC6 Q9UBN7 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9435428 0.90 ITGB3 (0.60) ITGB3ITGA2BCTSGCMA1HDAC1
SCHEMBL8776989 0.88 F2 (0.49) ITGB3ITGA2BF2F10PRSS1
SCHEMBL7387875 0.86 ITGB3 (0.76) ITGB3ITGA2BF2F10PRSS1
SCHEMBL7438806 0.83 ITGB3 (0.71) ITGB3ITGA2BPRSS1CTSGCMA1
Acetic Acid SCHEMBL9097876 0.82 ITGB3 (0.68) ITGB3ITGA2BPRSS1CTSGCMA1
SCHEMBL9710588 0.82 ITGB3 (0.64) ITGB3ITGA2BF2F10PRSS1
SCHEMBL7390380 0.82 ITGB3 (0.64) ITGB3ITGA2BF2F10PRSS1
Hydrochloric Acid SCHEMBL9435247 0.82 ITGB3 (0.70) ITGB3ITGA2BPRSS1CTSGCMA1
SCHEMBL9103107 0.82 ITGB3 (0.70) ITGB3ITGA2BPRSS1CTSGCMA1
SCHEMBL7386054 0.81 ITGB3 (0.76) ITGB3ITGA2BF2F10PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574545-B1 PHENYL AMIDINES DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 1994-11-30 EP claimed
US-6387880-B1 MIXTURE OF DRUG AND SOLVENT G.D. SEARLE & CO. 2002-05-14 US disclosed
EP-0729362-B1 TRANSDERMAL COMPOSITION OF N- N- 5- 4-(AMINOIMINOMETHYL)PHENYL]-1-OXOPENTYL]-L-alpha-ASPARTYL]-L-PHENYLALANINE OR ITS ESTERS AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS SEARLE & CO (US) 2000-01-12 EP disclosed
EP-0729362-A1 TRANSDERMAL COMPOSITION OF N- N- 5- 4-(AMINOIMINOMETHYL)PHENYL]-1-OXOPENTYL]-L-$g(a)-ASPARTYL]-L-PHENYLALANINE OR ITS ESTERS AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS G.D. SEARLE & CO. (US) 1996-09-04 EP disclosed
WO-1995013825-A1 TRANSDERMAL COMPOSITION OF N-[N-[5-[4-(AMINOIMINOMETHYL)PHENYL]-1-OXOPENTYL]-L-α-ASPARTYL]-L-PHENYLALANINE OR ITS ESTERS AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS G.D. SEARLE & CO. (US) 1995-05-26 WO disclosed