SCHEMBL7722111

SCHEMBL7722111

COC(=O)[C@@H]1C[C@@H](NC(=O)OC(C)(C)C)CN1C(=O)CN(C)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.38
MMP2 P08253 13/20 0.38
ANPEP P15144 6/20 0.36
CTSK P43235 2/20 0.36
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CYP2C9 P11712 1/20 0.34
HSD11B1 P28845 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7722109 1.00 BTK (0.38) BTKMMP2ANPEPCTSKCA1
SCHEMBL7727788 0.90 BTK (0.44) BTKMMP2ANPEPCTSKCA1
SCHEMBL7727791 0.90 BTK (0.44) BTKMMP2ANPEPCTSKCA1
SCHEMBL3103450 0.84 MMP2 (0.61) MMP2ANPEP
SCHEMBL2404149 0.84 MMP2 (0.61) MMP2ANPEP
SCHEMBL7731141 0.84 ALDH1A1 (0.43) MMP2ANPEPKMT2AALDH1A1
SCHEMBL7731145 0.84 ALDH1A1 (0.43) MMP2ANPEPKMT2AALDH1A1
SCHEMBL14467624 0.83 MMP2 (0.45) MMP2ANPEPKMT2AL3MBTL1
SCHEMBL7722292 0.83 ANPEP (0.52) MMP2ANPEPALDH1A1
SCHEMBL7722294 0.83 ANPEP (0.52) MMP2ANPEPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed
WO-2000001714-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed