SCHEMBL7723288

SCHEMBL7723288

O=C(C=CCNC1CCN(C[C@H]2CN([C@@H](CC3CCC3)C(=O)O)C[C@@H]2c2ccccc2)CC1)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.52
CACNA1F O60840 1/20 0.52
CACNA1D Q01668 1/20 0.52
CACNA1S Q13698 1/20 0.52
CACNA1C Q13936 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7730605 0.94 CCR5 (0.58) CCR5
SCHEMBL7723337 0.88 CCR5 (0.51) CCR5CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7732746 0.87 CCR5 (0.49) CCR5
SCHEMBL7730814 0.83 CCR5 (0.53) CCR5
SCHEMBL7733902 0.82 CCR5 (0.51) CCR5
SCHEMBL7736194 0.73 CCR5 (0.52) CCR5
SCHEMBL7730565 0.69 CCR5 (0.63) CCR5CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7541401 0.69 CCR5 (1.00) CCR5CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7492593 0.69 CCR5 (1.00) CCR5CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7987034 0.69 CCR5 (1.00) CCR5CACNA1FCACNA1DCACNA1SCACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399619-B1 PREVENTION AND TREATMENT OF AIDS AND VIRAL INFECTION BY HIV MERCK & CO., INC. 2002-06-04 US disclosed
WO-2000059497-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-10-12 WO disclosed