SCHEMBL7724496

SCHEMBL7724496

CCN(CC)N(c1ccccc1)S(=O)(=O)CC

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.44
ALDH1A1 P00352 1/20 0.44
GLA P06280 1/20 0.44
ESR1 P03372 3/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NR3C2 P08235 1/20 0.42
CA12 O43570 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
HSP90AA1 P07900 1/20 0.40
PSIP1 O75475 1/20 0.40
TP53 P04637 2/20 0.40
MAPT P10636 1/20 0.40
CNR2 P34972 2/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31357779 0.83 NR3C2 (0.46) TSHRALDH1A1GLAESR1MAPK1
SCHEMBL9779480 0.82 TSHR (0.47) TSHRALDH1A1GLAESR1MAPK1
SCHEMBL30872976 0.80 CA12 (0.50) TSHRALDH1A1GLAESR1MAPK1
SCHEMBL7920273 0.77 TSHR (0.41) TSHRALDH1A1GLAESR1MAPK1
SCHEMBL17333643 0.77 ESR1 (0.56) TSHRALDH1A1GLAESR1MAPK1
SCHEMBL4204976 0.76 PKM (0.47) TSHRALDH1A1GLAESR1MAPK1
SCHEMBL13762630 0.74 CA12 (0.50) TSHRALDH1A1GLAESR1MAPK1
SCHEMBL7645581 0.72 PSIP1 (0.41) TSHRALDH1A1GLAESR1MAPK1
SCHEMBL28347318 0.72 PSIP1 (0.41) TSHRALDH1A1GLAESR1MAPK1
SCHEMBL17333692 0.72 ESR1 (0.51) TSHRALDH1A1GLAESR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165514-A1 3-(ANILINOMETHYLENE) OXINDOLES AS PROTEIN TYROSINE KINASE AND PROTEIN SERINE/THREONINE KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2002-01-02 EP disclosed
WO-2000056710-A1 3-(ANILINOMETHYLENE) OXINDOLES AS PROTEIN TYROSINE KINASE AND PROTEIN SERINE/THREONINE KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2000-09-28 WO disclosed