SCHEMBL7727468

SCHEMBL7727468

O=C=Nc1cccc(Br)c1.O=C=Nc1cccc(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
MAPK1 P28482 1/20 0.38
MAOB P27338 2/20 0.37
IDO1 P14902 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 3/20 0.36
TRPA1 O75762 1/20 0.36
CTSL P07711 1/20 0.35
MEN1 O00255 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
RELA Q04206 1/20 0.34
GABRP O00591 2/20 0.33
GABRD O14764 2/20 0.33
GABRA1 P14867 2/20 0.33
GABRB1 P18505 2/20 0.33
GABRG2 P18507 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL59005 0.89 MAPK1 (0.45) KMT2ATDP1MAPK1IDO1ALDH1A1
SCHEMBL115285 0.89 NPC1 (0.46) KMT2ANPC1RAB9ATDP1MAPK1
SCHEMBL8589377 0.84 GABRA1 (0.40) KMT2ANPC1RAB9AMAOBIDO1
SCHEMBL8942928 0.82 NPC1 (0.45) KMT2ANPC1RAB9ATDP1MAPK1
SCHEMBL27912037 0.78 CYP3A4 (0.41) KMT2ANPC1RAB9ATDP1MAPK1
SCHEMBL8943320 0.77 CYP3A4 (0.42) KMT2ANPC1RAB9ATDP1MAPK1
SCHEMBL10615043 0.74 TDP1 (0.54) KMT2ANPC1RAB9ATDP1MAPK1
SCHEMBL27873 0.74 TDP1 (0.54) KMT2ANPC1RAB9ATDP1MAPK1
SCHEMBL29849778 0.74 TDP1 (0.39) KMT2ANPC1RAB9ATDP1MAPK1
SCHEMBL29849567 0.74 AGXT (0.40) TDP1MAPK1ALDH1A1CYP3A4TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015479-A4 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR LILLY CO ELI (US) 2002-07-24 EP disclosed
EP-1015479-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR ELI LILLY AND COMPANY (US) 2000-07-05 EP disclosed
WO-1998046631-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC MACROCYCLES AND PROCESSES THEREFOR ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed