SCHEMBL7729217

SCHEMBL7729217

CCN[C@@H](Cc1ccccc1)C(=O)OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.65
ATM Q13315 2/20 0.64
ALDH1A1 P00352 2/20 0.58
THRB P10828 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
HSD17B10 Q99714 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.57
TSHR P16473 1/20 0.56
GAA P10253 1/20 0.56
RAB9A P51151 1/20 0.56
CA12 O43570 1/20 0.55
CA2 P00918 1/20 0.55
CA7 P43166 1/20 0.55
CA9 Q16790 1/20 0.55
CA14 Q9ULX7 1/20 0.55
LMNA P02545 1/20 0.55
GLA P06280 1/20 0.55
ANPEP P15144 1/20 0.53
MEN1 O00255 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18435148 1.00 POLB (0.65) POLBATMALDH1A1THRBCYP2C9
SCHEMBL24925125 0.89 MMP8 (0.57) POLBATMALDH1A1L3MBTL1TSHR
SCHEMBL656070 0.89 MMP8 (0.57) POLBATMALDH1A1L3MBTL1TSHR
SCHEMBL25794712 0.87 POLB (0.51) POLBATMALDH1A1THRBCYP2C9
SCHEMBL7392765 0.87 POLB (0.70) POLBATMALDH1A1THRBCYP2C9
SCHEMBL9003236 0.87 POLB (0.70) POLBATMALDH1A1THRBCYP2C9
SCHEMBL20394526 0.87 TACR1 (0.56) POLBATMALDH1A1
SCHEMBL20394525 0.87 TACR1 (0.56) POLBATMALDH1A1
SCHEMBL7237658 0.87 ESR1 (0.59) POLBATMALDH1A1TSHRKMT2A
SCHEMBL19647162 0.87 ALDH1A1 (0.62) POLBATMALDH1A1THRBCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2861581-B9 1,2,3,4-Tetrahydroisoquinoline-pyrrolidine derivatives as antagonists of apoptosis (IAPs) for the treatment of cancer. BRISTOL MYERS SQUIBB CO (US) 2017-08-30 EP disclosed
US-8889712-B2 IAP antagonists BRISTOL-MYERS SQUIBB COMPANY (US) 2014-11-18 US disclosed
WO-2002083606-A1 A LINKER SYSTEM FOR THE SYNTHESIS AND SCREENING OF COMBINATORIAL LIBRARIES OF POLYAMINE DERIVATIVES ON WATER COMPATIBLE SUPPORTS UNIVERSITY OF ALBERTA (CA) 2002-10-24 WO disclosed