SCHEMBL7729772

SCHEMBL7729772

CCCn1c(=O)c2[nH]c(/C=C/c3ccccc3F)nc2n(CCC)c1=O

nearest known ligand 0.72

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 2/20 0.60
KDM4E B2RXH2 1/20 0.55
MEN1 O00255 1/20 0.55
ALDH1A1 P00352 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
ADORA2A P29274 1/20 0.55
CYP2C19 P33261 1/20 0.55
KMT2A Q03164 1/20 0.55
HSD17B10 Q99714 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7729777 1.00 ADORA2B (0.60) ADORA2BKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL7307763 0.90 ADORA2B (0.54) ADORA2BKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL7307772 0.90 ADORA2B (0.54) ADORA2BKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL7729464 0.87 KDM4E (0.55) ADORA2BKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL7729458 0.87 KDM4E (0.55) ADORA2BKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL7396871 0.84 KDM4E (0.62) ADORA2BKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL7396869 0.84 KDM4E (0.62) ADORA2BKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL8374185 0.81 KDM4E (0.53) ADORA2BKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL8374181 0.81 KDM4E (0.53) ADORA2BKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL7316340 0.81 ADORA2B (0.48) ADORA2BKDM4EALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628311-B1 Xanthine-Derivatives as Antidepressants KYOWA HAKKO KOGYO KK (JP) 2002-04-24 EP disclosed
EP-0565377-B1 Therapeutic agents for use in the treatment of Parkinson's Disease KYOWA HAKKO KOGYO KK (JP) 1998-01-07 EP disclosed
US-5587378-A ADMINISTERING A SUBSTITUTED XANTHINE COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-12-24 US disclosed
US-5543415-A ADMINISTERING A XANTHINE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-08-06 US disclosed
US-5484920-A XANTHINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-01-16 US disclosed
EP-0628311-A1 ANTIDEPRESSANT KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-12-14 EP disclosed
EP-0565377-A1 Therapeutic agents for use in the treatment of parkinson's disease KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-10-13 EP disclosed