SCHEMBL8374181

SCHEMBL8374181

CCCn1c(=O)c2[nH]c(/C=C/c3cccs3)nc2n(CCC)c1=O

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
ADORA2A P29274 1/20 0.53
ADORA2B P29275 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 1/20 0.53
HSD17B10 Q99714 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8374185 1.00 KDM4E (0.53) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL7396869 0.82 KDM4E (0.62) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL7396871 0.82 KDM4E (0.62) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL7729777 0.81 ADORA2B (0.60) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL7729772 0.81 ADORA2B (0.60) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL8373216 0.79 ADORA2A (0.52) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL7729464 0.79 KDM4E (0.55) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL7729458 0.79 KDM4E (0.55) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL8373214 0.79 ADORA2A (0.52) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL8371208 0.78 ADORA2B (0.55) ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559893-B1 XANTHINE DERIVATIVE KYOWA HAKKO KOGYO KK (JP) 1999-02-03 EP disclosed
US-5756735-A ADENOSINE A2 RECEPTOR ANTAGONISTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1998-05-26 US disclosed
EP-0559893-A1 XANTHINE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-15 EP disclosed