SCHEMBL7729803

SCHEMBL7729803

O=C(NC1CCN(CCc2ccccc2)C1)C1c2ccccc2Cc2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 1/20 0.56
SIGMAR1 Q99720 3/20 0.55
MC4R P32245 5/20 0.52
DRD4 P21917 3/20 0.47
DRD2 P14416 1/20 0.47
CXCR3 P49682 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
NAMPT P43490 1/20 0.45
HTR2A P28223 1/20 0.45
LTA4H P09960 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7729799 1.00 C3AR1 (0.56) C3AR1SIGMAR1MC4RDRD4DRD2
SCHEMBL7723289 0.91 C3AR1 (0.50) C3AR1SIGMAR1MC4RDRD4DRD2
SCHEMBL7723287 0.91 C3AR1 (0.50) C3AR1SIGMAR1MC4RDRD4DRD2
SCHEMBL7719821 0.85 CCR1 (0.62) SIGMAR1MC4RDRD4DRD2
SCHEMBL7719823 0.85 CCR1 (0.62) SIGMAR1MC4RDRD4DRD2
SCHEMBL7729609 0.85 SIGMAR1 (0.54) SIGMAR1MC4RDRD4DRD2CXCR3
SCHEMBL7724256 0.81 SIGMAR1 (0.57) SIGMAR1MC4RDRD4DRD2CXCR3
SCHEMBL7725101 0.80 SIGMAR1 (0.61) SIGMAR1MC4RDRD4DRD2CXCR3
SCHEMBL7725104 0.80 SIGMAR1 (0.61) SIGMAR1MC4RDRD4DRD2CXCR3
SCHEMBL7724247 0.79 SIGMAR1 (0.60) SIGMAR1MC4RDRD4DRD2CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6468998-B1 ANTAGONIZE SEROTONIN 2 RECEPTORS, SUPPRESS PLATELET AGGREGATION, IMPROVE PERIPHERAL CIRCULATION AND PROMOTE LACHRYMATION MITSUBISHI PHARMA CORPORATION (JP) 2002-10-22 US disclosed
EP-1125922-A1 PYRROLIDINE COMPOUNDS AND MEDICINAL UTILIZATION THEREOF Welfide Corporation (JP) 2001-08-22 EP disclosed