SCHEMBL7730376

SCHEMBL7730376

CCOC(=O)c1coc([C@@H](CCc2ccccc2)NC(=O)OC(C)(C)C)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.49
MAPT P10636 2/20 0.47
CTSK P43235 3/20 0.47
CTSS P25774 1/20 0.47
C3AR1 Q16581 1/20 0.46
ALDH1A1 P00352 5/20 0.45
CCR3 P51677 1/20 0.45
LMNA P02545 4/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
HSD17B10 Q99714 3/20 0.44
NPSR1 Q6W5P4 4/20 0.44
HPGD P15428 3/20 0.43
HTT P42858 3/20 0.43
XBP1 P17861 2/20 0.43
JAK2 O60674 1/20 0.43
S1PR4 O95977 1/20 0.43
HSP90AA1 P07900 1/20 0.43
THRB P10828 1/20 0.43
PKM P14618 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7723171 0.92 MAPT (0.56) TSHRMAPTCTSKCTSSC3AR1
SCHEMBL7735821 0.91 MAPT (0.47) TSHRMAPTCTSKCTSSC3AR1
SCHEMBL7723269 0.89 MAPT (0.48) TSHRMAPTCTSKCTSSC3AR1
SCHEMBL7733597 0.85 MAPT (0.51) TSHRMAPTCTSKCTSSC3AR1
SCHEMBL5014182 0.81 ALDH1A1 (0.56) TSHRMAPTCTSKCTSSC3AR1
SCHEMBL7861048 0.80 C3AR1 (0.44) TSHRMAPTCTSKCTSSC3AR1
SCHEMBL5014051 0.79 ALDH1A1 (0.58) TSHRMAPTCTSKCTSSC3AR1
SCHEMBL22648524 0.78 C3AR1 (0.47) TSHRMAPTCTSKCTSSC3AR1
SCHEMBL801072 0.78 PPARA (0.51) TSHRMAPTCTSSC3AR1ALDH1A1
Trifluoroacetic Acid SCHEMBL7735541 0.78 CCR3 (0.41) MAPTALDH1A1CCR3LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed